13th SCPA, ADVANCED ANALYTICAL METHODOLOGIES IN DRUG DISCOVERY
FINAL PROGRAM
September
21, 2008
14.00-19.00 Registration
15.00-18.15 Ph.D
thesis dissertations
18.15-18.45 Opening ceremony
18.45-19.30 Opening lecture: "MOLECULAR DEVICES
AND MACHINES" V. BALZANI
(University of Bologna, Italy)
19.30-20.30 Welcome
reception
September
22, 2008
PHARMACEUTICAL PROFILING ASSAYS IN DRUG DISCOVERY:
NEW ANALYTICAL APPROACHES
9.00-9.30
Opening
of the 13th SCPA (V. ANDRISANO)
Chairman:
S. Pinzauti (University of Firenze, Italy)
9.30-11.00
‘NEW HTS ASSAYS TO STUDY LIPOPHYLICITY, pKa AND PERMEABILITY
OF DRUG-LIKE COMPOUNDS.’ S. MARTEL and
J-L VEUTHEY (Université de Genève, Switzerland)
11.00-11.15
Coffee break
11.15-12.15
"SOLUBILITY ASSESSMENT IN DRUG DISCOVERY" S. BEATO
(GSK, Verona, Italy)
12.15-13.30
Lunch
Chairman:
G. Massolini (University
of Pavia, Italy)
13.30-14.15
"STRATEGIES AND METHODS FOR ASSESSING BLOOD-BRAIN-BARRIER PENETRATION
IN THE DRUG DISCOVERY PROCESS" G. WESTERBERG (SienaBiotech,
Siena, Italy)
14.30-15.30
"DYNAMIC LIGHT SCATTERING AGGREGATION STUDIES" D.
FRISCIONE (Alphatech, Genova, Italy).
15.30-15.45
Coffee break
15.45-17.15
"TUTORIALS IN THE INFORMATIC ROOM FOR PHYSICO-CHEMICAL PARAMETERS
DETERMINATION". S. MARTEL (Université
de Genève, Switzerland)
17.15-18.15
"TUTORIALS IN THE INFORMATIC ROOM FOR LIGHT SCATTERING APPLICATIONS".
D. FRISCIONE (Alphatech, Genova, Italy).
September
23, 2008
HIT IDENTIFICATION: ADVANCES IN ANALYTICAL
METHODS
Chairman:
C. Bertucci (University of Bologna, Italy)
9.00-9.30
“BIOANALYSIS IN DRUG DISCOVERY: AN INTRODUCTION” G.
ALDINI (Istituto di Chimica Farmaceutica e Tossicologica
"Pietro Pratesi", University of Milan, Italy)
9.30-10.30
“BIOPHYSICAL TOOLS FOR STUDYING BIOMOLECULAR INTERACTIONS
- FRAGMENT-BASED APPROACHES IN DRUG DISCOVERY” A.
PADOVA (SienaBiotech, Siena, Italy).
10.30-10.45
Coffee break
10.45-12.45
“CIRCULAR DICHROISM: DRUG DISCOVERY AND DRUG DESIGN”
A. F. DRAKE (Department of Pharmacy, King's College,
London).
12.45-14.00
Lunch
Chairman:
J.-L.
Veuthey (Université de Genève, Switzerland)
14.00-15.00
“HIT SELECTION BY CAPILLARY ELECTROPHORESIS” E.
DE LORENZI (Department of Pharmaceutical Chemistry, University
of Pavia, Italy).
15.00–16.00
"OPTICAL BIOSENSORS AS TOOLS FOR DRUG DISCOVERY” H.
DANIELSON (Department of Biochemistry, Uppsala University,
Sweden).
16.00-16.15
Coffee break
16:15-17:30
"TUTORIALS IN THE INFORMATIC ROOM ON APPLICATION AND ANALYSIS
BY BIOSENSORS". H. DANIELSON (Department of
Biochemistry, Uppsala University, Sweden)
17.30
Closure of the 13th SCPA
20.00 Social dinner
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